富山県立大学工学部 医薬品工学科 バイオ医薬品工学講座

安田研究室

                                                      

2019

2019年

  1. Sulfate conjugates are the major metabolites in rats administrated with sesamin.
    Yasuda K, Okamoto K, Ueno S, Itoh K, Nishikawa M, Ikushiro S, Sakaki T.
    Drug Metab Pharmacokinet. 34(2):134-140 (2019)


  2. Introduction of fluorine atoms to vitamin D3 side-chain and synthesis of 24,24-difluoro-25-hydroxyvitamin D3.
    Kawagoe F, Mototani S, Yasuda K, Nagasawa K, Uesugi M, Sakaki T, Kittaka A.
    J Steroid Biochem Mol Biol. 195:105477. doi: 10.1016/j.jsbmb.2019.105477. (2019)


  3. Synthesis and CYP24A1-Dependent Metabolism of 23-Fluorinated Vitamin D3 Analogues.
    Kawagoe F, Yasuda K, Mototani S, Sugiyama T, Uesugi M, Sakaki T, Kittaka A.
    ACS Omega. 4: 11332-11337. (2019)


  4. Membrane fusogenic high-density lipoprotein nanoparticles
    Kim H, Nobeyama T, Honda S, Yasuda K, Morone N, Murakami T.
    Biochim Biophys Acta Biomembr. 1861(10): 183008. (2019)


  5. Dimethyl fumarate and vitamin D derivatives cooperatively enhance VDR and Nrf2 signaling in differentiating AML cells in vitro and inhibit leukemia progression in a xenograft mouse model.
    Nachliely M, Trachtenberg A, Khalfin B, Nalbandyan K, Cohen-Lahav M, Yasuda K, Sakaki T, Kutner A, Danilenko M.
    J Steroid Biochem Mol Biol. 188:8-16 (2019)


  6. Concise synthesis of 23-hydroxylated vitamin D3 metabolites.
    Kawagoe F, Sugiyama T, Yasuda K, Uesugi M, Sakaki T, Kittaka A.
    J Steroid Biochem Mol Biol. 186:161-168. (2019).


メニュー

コンテンツへスキップ
  • トップページ

Copyright ©富山県立大学工学部 医薬品工学科 バイオ医薬品工学講座安田研究室 , All rights reserved.